PCS1055, CAS [[357173-55-8]]

Produktübersicht

• Artikelname: PCS1055, CAS [[357173-55-8]]
• Artikelnummer: TGM-T88610
• Hersteller Artikelnummer: T88610
• Alternativnummer: TGM-T88610-25MG,TGM-T88610-50MG,TGM-T88610-100MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien

Produktbeschreibung

PCS1055 is a selective and competitive antagonist of the muscarinic M4 receptor (muscarinic M4 receptor), with an IC50 of 18.1 nM and a Kd of 5.72 nM. It inhibits the binding of the radioligand [3H]-NMS to the M4 receptor, with a Ki of 6.5 nM. Additionally, PCS1055 acts as an AChE inhibitor, exhibiting IC50 values of 22 nM for electric eel AChE and 120 nM for human AChE.

Produkteigenschaften

• Molekulargewicht: 412.57
• CAS Nummer: [357173-55-8]
• Formel: C27H32N4
• Target-Kategorie: Cholinesterase (ChE)|||AChR

Bilder

T88610