PCS1055 is a selective and competitive antagonist of the muscarinic M4 receptor (muscarinic M4 receptor), with an IC50 of 18.1 nM and a Kd of 5.72 nM. It inhibits the binding of the radioligand [3H]-NMS to the M4 receptor, with a Ki of 6.5 nM. Additionally, PCS1055 acts as an AChE inhibitor, exhibiting IC50 values of 22 nM for electric eel AChE and 120 nM for human AChE.
Molecular Weight:
412.57
CAS Number:
[357173-55-8]
Formula:
C27H32N4
Target:
Cholinesterase (ChE)|||AChR
T88610
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