IGF-1Rmodulator 1 (Example 5) is an IGF-1R modulator featuring an EC50 of 0.29 µM (FGFR1), 0.25 µM (IGF1R), 0.34 µM (TrkA), and 0.39 µM (TrkB). This compound is useful in research on diseases characterized by impaired signaling of neurotrophic and/or other trophic factors, such as Alzheimers disease.
Molekulargewicht:
387.39
CAS Nummer:
[2375424-89-6]
Formel:
C22H17N3O4
Target-Kategorie:
EGFR|||Trk receptor|||IGF-1R
T88615
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