PF-04802367, CAS [[1962178-27-3]]

Artikelnummer: TGM-T9611
Artikelname: PF-04802367, CAS [[1962178-27-3]]
Artikelnummer: TGM-T9611
Hersteller Artikelnummer: T9611
Alternativnummer: TGM-T9611-1MLX10MM(INDMSO),TGM-T9611-1MG,TGM-T9611-5MG,TGM-T9611-10MG,TGM-T9611-25MG,TGM-T9611-50MG,TGM-T9611-100MG,TGM-T9611-200MG
Hersteller: TargetMol
Kategorie: Biochemikalien
PF-04802367 is a highly selective GSK-3 inhibitor with an IC50 of 2.1 nM based on a recombinant human GSK-3beta enzyme assay and 1.1 nM based on ADP-Glo assay. It shows desirable central nervous system (CNS) properties and potency. It is equally effective at inhibition of the two known GSK-3 isoforms (GSK-3alpha and GSK-3beta) with IC50 values of 10.0 and 9.0 nM in mobility shift assays, respectively.
Molekulargewicht: 361.78
Reinheit: 98.76%
CAS Nummer: [1962178-27-3]
Formel: C16H16ClN5O3
Target-Kategorie: GSK-3
T9611