Opiranserin hydrochloride, CAS [[1440796-75-7]]

Artikelnummer: TGM-T9833
Artikelname: Opiranserin hydrochloride, CAS [[1440796-75-7]]
Artikelnummer: TGM-T9833
Hersteller Artikelnummer: T9833
Alternativnummer: TGM-T9833-1MLX10MM(INDMSO),TGM-T9833-1MG,TGM-T9833-5MG,TGM-T9833-10MG,TGM-T9833-25MG,TGM-T9833-50MG,TGM-T9833-100MG,TGM-T9833-500MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 µM, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 µM). It is development as an injectable agent for the treatment of postoperative pain.
Molekulargewicht: 430.97
Reinheit: 99.33%
CAS Nummer: [1440796-75-7]
Formel: C21H35ClN2O5
Target-Kategorie: GlyT|||5-HT Receptor|||P2X Receptor
T9833