4,5-Dimethoxycanthin-6-one, CAS [[18110-87-7]]

Produktübersicht

• Artikelname: 4,5-Dimethoxycanthin-6-one, CAS [[18110-87-7]]
• Artikelnummer: TGM-TN3013
• Hersteller Artikelnummer: TN3013
• Alternativnummer: TGM-TN3013-1MLX10MM(INDMSO), TGM-TN3013-1MG, TGM-TN3013-5MG, TGM-TN3013-10MG, TGM-TN3013-25MG, TGM-TN3013-50MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien
• Alternative Synonym: Methylnigakinone

Produktbeschreibung

4,5-Dimethoxycanthin-6-one is an alkaloid isolated from Picrasma quassioides BENNET (Simaroubaceae) with antimicrobial activity against Staphylococcus aureus and its drug-resistant strains. It is a potent, non-competitive inhibitor of CYP1A2-mediated phenacetin O-deethylation (IC50: 1.7 µM, Ki: 2.6 µM) and a potent inhibitor of cyclic adenosine monophosphate (cAMP) phosphodiesterase. Additionally, it exhibits cytotoxicity to tumor cell lines U937 and HepG2.

Produkteigenschaften

• Molekulargewicht: 280.28
• Reinheit: 0.9893
• CAS Nummer: [18110-87-7]
• Formel: C16H12N2O3
• Target-Kategorie: PDE|||Cytochromes P450|||Antibacterial