CCT036477 is an inhibitor of Wnt signaling. Studies show that CCT036477 does not alter beta-catenin levels but blocks transcription at the beta-catenin level. CCT036477 inhibited growth in several cancer cell lines and showed clear activity in vivo, blocking development of Zebrafish and Xenopus embryos and expression of Wnt target genes.
Molekulargewicht:
347.84
CAS Nummer:
[305372-78-5]
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