CC-90011 (Pulrodemstat) benzenesulfonate is a potent, selective, reversible and orally active lysine-specific demethylase-1 (LSD1) inhibitor,IC50 0.25 nM. CC-90011 benzenesulfonate has less enzymatic inhibition of LSD2, MOA-A and MAO-B. CC-90011 benzenesulfonate induces differentiation of acute myeloid leukemia (AML) and small cell lung cancer (SCLC) cells and has potent anti-cancer activity.
Molecular Weight:
609.65
Purity:
>99%
CAS Number:
[2097523-60-7]
Formula:
C30H29F2N5O5S
Target:
Histone demethylase
* VAT and and shipping costs not included. Errors and price changes excepted