BMS-986158 is a potent BET inhibitor with IC50s of 6.6 and 5 nM in NCI-H211 small cell lung cancer (SCLC) cells and MDA-MB231 triple negative breast cancer (TNBC) cells, respectively.
Molecular Weight:
495.62
Purity:
>99%
CAS Number:
[1800340-40-2]
Target:
Epigenetic Reader Domain
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