TAK-243 (MLN7243) is a first-in-class, selective ubiquitin activating enzyme, UAE (UBA1) inhibitor (IC50=1 nM), which blocks ubiquitin conjugation, disrupting monoubiquitin signaling as well as global protein ubiquitination.
Molecular Weight:
519.52
Purity:
>98%
CAS Number:
[1450833-55-2]
Target:
E1/E2/E3 Enzyme
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