Mozavaptan (OPC-31260) is a benzazepine derivative and a potent, selective, competitive and orally active vasopressin V2 receptor antagonist with an IC50 of 14 nM. Mozavaptan shows ~85-fold selectivity for V2 receptor over V1 receptor (IC50 of 1.2 µM), and can antagonize the antidiuretic action of arginine vasopressin (AVP) in vivo.
Molecular Weight:
427.53
Purity:
99.12%
CAS Number:
[137975-06-5]
Formula:
C27H29N3O2
Target:
Vasopressin Receptor
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