Loperamide hydrochloride is a high affinity µ-opioid receptor agonist with peripheral selectivity with Ki values of 2, 48 and 1156 nM for µ-, delta- and kappa-opioid receptors respectively. Loperamide hydrochloride is also a selective and competitive human intestinal carboxylesterases (hiCE) inhibitor. It can be used to construct animal models of functional constipation.
Molecular Weight:
513.51
Purity:
100.0%
CAS Number:
[34552-83-5]
Formula:
C29H33ClN2O2.HCl
Target:
Animal Modeling
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