Epoxomicin (BU-4061T) is a cell-permeable, selective and irreversible proteasome inhibitor with an IC50 value of 4 nM. Epoxomicin covalently binds to the LMP7, X, MECL1, and Z catalytic subunits of the proteasome and potently inhibits primarily the chymotrypsin-like activity. Epoxomicin can cross the blood-brain barrier.
Molecular Weight:
554.72
Purity:
>99.0%
CAS Number:
[134381-21-8]
Formula:
C28H50N4O7
Target:
Proteasome
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