Agomelatine is a metabolically stable analog of melatonin that displays agonist activity for MT1 and MT2 binding with nanomolar affinity. Agomelatine is also a selective 5-HT2C receptor antagonist with pKis of 6.4 and 6.2 at native (porcine) and cloned, human 5-HT2C receptors, respectively.
Molecular Weight:
243.3
Purity:
99.93%
CAS Number:
[138112-76-2]
Formula:
C15H17NO2
Target:
Melatonin Receptor
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