Adapalene is a third-generation topical retinoid, it is a potent RAR agonist, with AC50 values of 2.3 nM, 9.3 nM, and 22 nM for RARbeta, RARgamma, RARalpha, respectively. Adapalene also inhibits the enzymatic activity of GOT1 in a non-competitive manner. Adapalene is also an MST1 agonist.
Molecular Weight:
412.52
Purity:
>99%
CAS Number:
[106685-40-9]
Formula:
C28H28O3
Target:
RAR/RXR
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