ERG240 is a selective inhibitor of branched-chain aminotransferase 1 (BCAT1) with an IC50 of 0.1-1nM. ERG240 leads to decreased oxygen consumption and glycolysis through the down regulation of IRG1 expression, which leads to decrease itaconate production in human macrophages.
Molecular Weight:
166.15
Purity:
>98.5%
CAS Number:
[1415683-79-2]
Formula:
C7H11NaO3
Target:
Transferase
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