Linopirdine (DuP 996) is an orally active, selective M-type K+ current (IM, Kv7, KCNQ Channels) inhibitor with an IC50 of 2.4 µM. Linopirdine is a TRPV1 agonist. Linopirdine, a putative cognition enhancing agent, increases acetylcholine release in rat brain tissue.
Molecular Weight:
391.46
Purity:
99.0%
CAS Number:
[105431-72-9]
Formula:
C26H21N3O
Target:
Potassium Channel
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