Endoxifen Z-isomer is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERalpha). Endoxifen inhibits hERG tail currents at 50 mV in a concentration-dependent manner with IC50 values of 1.6 µM.
Molecular Weight:
373.49
Purity:
99.0%
CAS Number:
[112093-28-4]
Formula:
C25H27NO2
Target:
Estrogen Receptor
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