GDC-0276 is a potent, selective, reversible and orally active NaV1.7 inhibitor with an IC50 value of 0.4 nM. GDC-0276 is well tolerated and exhibits a good pharmacokinetic profile. GDC-0276 has the potential for the treatment of pain and to address shortcomings of existing pain medications, such as addiction and off-target side effects.
Molecular Weight:
462.58
Purity:
99.0%
CAS Number:
[1494581-70-2]
Formula:
C24H31FN2O4S
Target:
Sodium Channel
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