PU139 is a potent pan-histone acetyltransferase (HAT) inhibitor. PU139 blocks the HATs Gcn5, p300/CBP-associated factor (PCAF), CREB (cAMP response element-binding) protein (CBP) and p300 with IC50s of 8.39, 9.74, 2.49 and 5.35 µM, respectively.
Molecular Weight:
246.26
Purity:
99.0%
CAS Number:
[158093-65-3]
Formula:
C12H7FN2OS
Target:
Histone Acetyltransferase
* VAT and and shipping costs not included. Errors and price changes excepted