Pentoxyverine citrate is an orally active sigma-1 receptor agonist with Ki values of 41 nM for sigma1, 894 nM for sigma2, and 75 nM for sigma1 in guinea pig brain membranes.Pentoxyverine citrate is also a muscarinic antagonist.
Molecular Weight:
525.59
Purity:
>98%
CAS Number:
[23142-01-0]
Formula:
C20H31NO3.C6H8O7
Target:
Sigma Receptor
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