ARP-100 is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM). ARP-100 interacts with S1 pocket of MMP-2 and shows anti-invasive properties in an in vitro model of invasion on matrigel. ARP-100 shows the less inhibitory activity towards MMP-1 (>50 µM), MMP-3 (4.5 µM), MMP-7 (>50 µM), and MMP-9 (0.2 µM).
Molecular Weight:
364.42
Purity:
99.0%
CAS Number:
[704888-90-4]
Formula:
C17H20N2O5S
Target:
MMP
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