PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
Molecular Weight:
499.52
Purity:
>98%
CAS Number:
[1627676-59-8]
Formula:
C23H25F4N3O3S
Target:
Histone Methyltransferase
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