Serabelisib (INK-1117,MLN-1117,TAK-117) is a potent and selective oral PI3Kalpha isoform inhibitor (IC50 of 21 nmol/L against PI3Kalpha) that has demonstrated > 100-fold selectivity relative to other class I PI3K family members (PI3Kbeta/gamma/delta) and mTOR, and a high degree of selectivity against many other kinase.
Molecular Weight:
363.37
Purity:
>99.0%
CAS Number:
[1268454-23-4]
Formula:
C19H17N5O3
Target:
PI3K
* VAT and and shipping costs not included. Errors and price changes excepted