AR-C 118925XX is a selective, competitive P2Y2 receptor antagonist. AR-C 118925XX is inactive against a panel of 37 other receptors at a concentration of 10 µM. AR-C 118925XX inhibits ATP-gammaS-induced mucin secretion in bronchial epithelial cells (IC50 = 1 µM). AR-C 118925XX inhibits P2Y2 receptor-induced beta-arrestin translocation in vitro (pA2 = 37.2-51.3 nM).
Molecular Weight:
537.59
Purity:
>98%
CAS Number:
[216657-60-2]
Formula:
C28H23N7O3S
Target:
P2 Receptor
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