Lestaurtinib is a potent JAK2, FLT3 and TrkA inhibitor (IC50 values are 0.9, 3 and < 25 nM, respectively). Lestaurtinib also inhibits Aurora kinase A and B (IC50 values are 8.1 and 2.3 nM, respectively) and prevents STAT5 phosphorylation (IC50 = 20 - 30 nM).
Molecular Weight:
439.46
Purity:
99.0%
CAS Number:
[111358-88-4]
Formula:
C26H21N3O4
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