ML221 is an Apelin (APJ) antagonist and inhibits apelin-13-mediated activation of APJ. IC50 values of cAMP and beta -Arrestin were 0.70 µM and 1.75 µM, respectively. EC80 values were all 10 nM.
Molecular Weight:
385.35
Purity:
99.0%
CAS Number:
[877636-42-5]
Formula:
C17H11N3O6S
Target:
Apelin Receptor
* VAT and and shipping costs not included. Errors and price changes excepted