UK-78282 is a novel, potent and selective Kv1.3 blocker with an IC50 of 200 nM. UK-78282 effectively suppresses human T-lymphocyte activation in vitro. UK-78282 binds to residues at the inner surface of the channel overlapping the site of action of verapamil.
Molecular Weight:
466.05
Purity:
99.0%
CAS Number:
[136647-02-4]
Formula:
C29H35NO2HCl
Target:
Potassium Channel
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