OICR9429 --- WDR5 Antagonist, CAS [[1801787-56-3]], Unconjugated

Product Overview

• Article Name: OICR9429 --- WDR5 Antagonist, CAS [[1801787-56-3]], Unconjugated
• Biozol Catalog Number: BSS-BS-60255C
• Supplier Catalog Number: bs-60255C
• Alternative Catalog Number: BSS-BS-60255C-10,BSS-BS-60255C-2
• Manufacturer: Bioss
• Category: Biochemikalien
• Conjugation: Unconjugated

Product Description

OICR9429 is a potent and selective WD repeat-containing protein 5 (WDR5) antagonist (Kd ~24-52 nM). It has >100-fold selectivity over other methyltransferases tested. It disrupts WDR5 interaction with peptide regions of MLL and Histone 3. OICR-9429 also disrupts the interaction of WDR5 with MLL1 and RbBP5 in cells with IC50 values below 1 µM.

Product Properties

• Buffer: Powder
• CAS Number: [1801787-56-3]