SSR240612 is a potent and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors respectively).
Molecular Weight:
793.4
Purity:
>98% (HPLC)
CAS Number:
[464930-42-5]
Formula:
C42H53ClN4O7S
Target:
B1 Receptor
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