PIK-75 Hydrochloride is a p110alpha inhibitor with IC50 of 5.8 nM (200-fold more potently than p110beta), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM in cell-free assays.
Molecular Weight:
452.3
Purity:
>98% (HPLC)
CAS Number:
[372196-67-3]
Formula:
C16H14BrN5O4S
Target:
DNA-PK| p110alpha| p110beta| p110gamma| p110delta
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