ETP-46321 is a potent, orally active small molecule inhibitor targeting PI3Kalpha and PI3Kdelta isoforms with Kis of 2.3 nM and 14.2 nM, respectively. It is a valuable research tool for investigating PI3K signaling in oncology and immunology, supporting both in vitro cellular assays and in vivo pharmacokinetic and efficacy studies.
Molecular Weight:
473.55
Purity:
99.80% (May vary between batches)
CAS Number:
[1252594-99-2]
Formula:
C20H27N9O3S
Target:
PI3K
Application Notes:
Solubility: DMSO:30 mg/mL (63.35 mM)
* VAT and and shipping costs not included. Errors and price changes excepted