This compound is a highly selective and potent agonist of the NK2 receptor, exhibiting an IC50 of 6.1 nM. It effectively induces smooth muscle contraction in isolated rat fundus and bladder tissues, with EC50 values of 117 nM and 10 nM, respectively. This makes it a valuable research tool for studying tachykinin receptor function in gastrointestinal and urogenital systems.
Molecular Weight:
803.99
Purity:
>99.99% (May vary between batches)
CAS Number:
[137565-28-7]
Formula:
C39H65N9O9
Target:
Neurokinin receptor
Application Notes:
Solubility: H2O:1 mg/mL (1.24 mM)
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