Neurokinin receptor, Neurokinin Receptor, Neurokininreceptor, NK receptor, NK1, inhibit, Inhibitor, GR73632, GR-73632, GR 73632, Tachykinin receptor
This small molecule is a potent and selective agonist of the neurokinin 1 (NK1) receptor, exhibiting an EC50 of 2 nM in the guinea pig vas deferens assay. It is a valuable research tool for investigating the role of substance P signaling in pain, inflammation, and emesis through both in vitro and in vivo experimental models.