GSK620, CAS [[2088410-46-0]]

Product Overview

• Article Name: GSK620, CAS [[2088410-46-0]]
• Biozol Catalog Number: BYT-ORB1298440
• Supplier Catalog Number: orb1298440
• Alternative Catalog Number: BYT-ORB1298440-1, BYT-ORB1298440-10, BYT-ORB1298440-100, BYT-ORB1298440-2, BYT-ORB1298440-200, BYT-ORB1298440-25, BYT-ORB1298440-5, BYT-ORB1298440-50
• Manufacturer: Biorbyt
• Category: Biochemikalien
• Alternative Names: anti-inflammatory, blood, human, GSK 620, GSK620, GSK-620, EpigeneticReaderDomain, Epigenetic Reader Domain, oral, pan-BD2, inhibit, Inhibitor, phenotype, whole, selectivity

Product Description

GSK620 is a highly selective pan-BD2 BET inhibitor demonstrating potent anti-inflammatory activity in human whole blood assays. Its excellent selectivity profile and favorable oral pharmacokinetics support its use for in vivo research into inflammation and oncology, where BET bromodomain function is implicated.

Product Properties

• Molecular Weight: 325.36
• Purity: 99.88% (May vary between batches)
• CAS Number: [2088410-46-0]
• Formula: C18H19N3O3
• Target: Epigenetic Reader Domain

Application Notes

• Application Notes: Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (10.14 mM),DMSO:45 mg/mL (138.31 mM)