CPI-169 racemate, CAS [[1450655-76-1]]

Product Overview

• Article Name: CPI-169 racemate, CAS [[1450655-76-1]]
• Biozol Catalog Number: BYT-ORB1300447
• Supplier Catalog Number: orb1300447
• Alternative Catalog Number: BYT-ORB1300447-1,BYT-ORB1300447-2,BYT-ORB1300447-5,BYT-ORB1300447-10,BYT-ORB1300447-25,BYT-ORB1300447-50,BYT-ORB1300447-100
• Manufacturer: Biorbyt
• Category: Biochemikalien
• Alternative Names: CPI 169, CPI 169 racemate, CPI169, CPI-169, CPI169 racemate, CPI-169 racemate, EZH1, EZH2 WT, EZH2 Y641N, Epigenetic Reader Domain, EpigeneticReaderDomain, Histone Methyltransferase, HistoneMethyltransferase

Product Description

CPI-169 is a highly potent and selective inhibitor of EZH2, demonstrating IC50 values of 0.24 nM for wild-type, 0.51 nM for the Y641N mutant, and 6.1 nM for EZH1. This compound is a valuable chemical probe for epigenetic research, enabling the study of histone methylation roles in cancer biology and other diseases in both cellular and animal models.

Product Properties

• Molecular Weight: 528.66
• Purity: 99.59% (May vary between batches)
• CAS Number: [1450655-76-1]
• Formula: C27H36N4O5S
• Target: Epigenetic Reader Domain,Histone Methyltransferase

Application Notes

• Application Notes: Solubility: Ethanol:93 mg/mL (175.92 mM),H2O:< 1 mg/mL (insoluble or slightly soluble),DMSO:93 mg/mL (175.92 mM)