inhibit, KAD 1229, KAD1229, KAD-1229, KcsA, Mitiglinide, Mitiglinide Calcium, insulinotropic, Inhibitor, hypoglycaemic, diabetes, ATP-sensitive K+ channels, anti-diabetic, S-21403, S21403, S 21403, Potassium Channel, PotassiumChannel, type
Mitiglinide Calcium (KAD-1229) is a rapid-acting insulin secretagogue that functions by blocking ATP-sensitive potassium channels in pancreatic beta-cells. It is a valuable research tool for studying glucose homeostasis and insulin secretion mechanisms in both in vitro cellular assays and in vivo models of type 2 diabetes.
Molecular Weight:
668.88
Purity:
99.83% (May vary between batches)
CAS Number:
[145525-41-3]
Formula:
(C19H24NO3)2Ca
Target:
Potassium Channel,ATPase
Application Notes:
Solubility: DMSO:5 mg/mL (7.48 mM)
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