GW842166X is a potent and selective CB2 receptor agonist (EC50 = 63 nM) with negligible activity at CB1. It has been investigated in Phase 2 clinical trials and is a valuable research tool for studying CB2 function in inflammatory and neuropathic pain models, both in vitro and in vivo.
Molecular Weight:
449.25
Purity:
99.88% (May vary between batches)
CAS Number:
[666260-75-9]
Formula:
C18H17Cl2F3N4O2
Target:
Cannabinoid Receptor
Application Notes:
Solubility: H2O:< 1 mg/mL (insoluble or slightly soluble),DMSO:16 mg/mL (35.61 mM),Ethanol:< 1 mg/mL (insoluble or slightly soluble)
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