Galeterone, CAS [[851983-85-2]]

Product Overview

• Article Name: Galeterone, CAS [[851983-85-2]]
• Biozol Catalog Number: BYT-ORB1300706
• Supplier Catalog Number: orb1300706
• Alternative Catalog Number: BYT-ORB1300706-1, BYT-ORB1300706-10, BYT-ORB1300706-100, BYT-ORB1300706-200, BYT-ORB1300706-25, BYT-ORB1300706-5, BYT-ORB1300706-50
• Manufacturer: Biorbyt
• Category: Biochemikalien
• Alternative Names: Inhibitor, Galeterone, inhibit, AndrogenReceptor, Androgen Receptor, CYPs, CYP17, Cytochrome P450, TOK 001, TOK001, TOK-001, VN 124, VN/124-1, VN124, VN-124, VN-124-1

Product Description

Galeterone (VN 124) is an orally active small molecule that antagonizes the androgen receptor, inhibits CYP17A1 lyase activity, and reduces androgen receptor protein levels, thereby suppressing androgen signaling in prostate cancer. It is used in research for studying castration-resistant prostate cancer mechanisms and has been evaluated in both in vitro assays and in vivo xenograft models.

Product Properties

• Molecular Weight: 388.55
• Purity: 99.77% (May vary between batches)
• CAS Number: [851983-85-2]
• Formula: C26H32N2O
• Target: Cytochromes P450,Androgen Receptor

Application Notes

• Application Notes: Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.15 mM),DMSO:19.4 mg/mL (49.93 mM),Ethanol:19.4 mg/mL (49.93 mM)