SSR240612, CAS [[464930-42-5]]

Product Overview

• Article Name: SSR240612, CAS [[464930-42-5]]
• Biozol Catalog Number: BYT-ORB1302140
• Supplier Catalog Number: orb1302140
• Alternative Catalog Number: BYT-ORB1302140-1, BYT-ORB1302140-5, BYT-ORB1302140-1, BYT-ORB1302140-10, BYT-ORB1302140-25, BYT-ORB1302140-50, BYT-ORB1302140-100
• Manufacturer: Biorbyt
• Category: Biochemikalien
• Alternative Names: SSR 240612, SSR240612, SSR-240612, Inhibitor, inhibit, B1 Receptor, BradykininReceptor, Bradykinin Receptor

Product Description

SSR240612 is a potent, orally bioavailable non-peptide antagonist that selectively targets the bradykinin B1 receptor, demonstrating high affinity (Ki = 0.48-0.73 nM) and excellent selectivity over the B2 receptor. It is a valuable research tool for investigating the role of the B1 receptor in pain, inflammation, and neuropathic conditions in both in vitro and in vivo models.

Product Properties

• Molecular Weight: 793.41
• Purity: 99.16% (May vary between batches)
• CAS Number: [464930-42-5]
• Formula: C42H53ClN4O7S
• Target: Bradykinin Receptor

Application Notes

• Application Notes: Solubility: H2O:Insoluble,10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (5.04 mM),DMSO:100 mg/mL (126.04 mM)