BAR 501, BAR501, BAR-501, G-protein coupled receptor 19, G protein-coupled Bile Acid Receptor 1, GPBAR1, GPCR19, inhibit, Inhibitor, TGR5
BAR501 is a potent and selective agonist for the GPBAR1 receptor, exhibiting an EC50 of 1 µM. This small molecule is a valuable research tool for investigating GPBAR1s role in metabolic and inflammatory pathways, applicable in both in vitro and in vivo experimental models.