CPI-360, CAS [[1802175-06-9]]

Product Overview

• Article Name: CPI-360, CAS [[1802175-06-9]]
• Biozol Catalog Number: BYT-ORB1685548
• Supplier Catalog Number: orb1685548
• Alternative Catalog Number: BYT-ORB1685548-1, BYT-ORB1685548-10, BYT-ORB1685548-100, BYT-ORB1685548-25, BYT-ORB1685548-5, BYT-ORB1685548-50
• Manufacturer: Biorbyt
• Category: Biochemikalien
• Alternative Names: Synonym 2, Synonym 2, Histone Methyltransferase, HistoneMethyltransferase, EZH2, CPI 360, CPI360, CPI-360, Apoptosis

Product Description

CPI-360 is a potent and selective small molecule inhibitor of EZH2, demonstrating sub-nanomolar enzymatic inhibition and cellular activity. It has shown antitumor efficacy in EZH2-dependent xenograft models, supporting its use as a chemical probe for epigenetic research in oncology, both in vitro and in vivo.

Product Properties

• Molecular Weight: 437.53
• Purity: 99.89% (May vary between batches)
• CAS Number: [1802175-06-9]
• Formula: C25H31N3O4
• Target: Apoptosis,Histone Methyltransferase

Application Notes

• Application Notes: Solubility: H2O:< 1 mg/mL (insoluble or slightly soluble),DMF:9 mg/mL (20.57 mM),Ethanol:27 mg/mL (61.71 mM),DMSO:22.5 mg/mL (51.43 mM)