M-808 is a potent, covalent small-molecule inhibitor that disrupts the Menin-MLL protein-protein interaction with high affinity (IC50 = 2.6 nM). It is a valuable chemical probe for researching MLL-rearranged leukemias and has demonstrated utility in both in vitro biochemical assays and in vivo xenograft models.
Molecular Weight:
819.09
CAS Number:
[2377335-74-3]
Formula:
C45H63FN6O5S
Target:
Others,Epigenetic Reader Domain
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