Apinocaltamide, CAS [[1838651-58-3]]

Product Overview

• Article Name: Apinocaltamide, CAS [[1838651-58-3]]
• Biozol Catalog Number: BYT-ORB1707717
• Supplier Catalog Number: orb1707717
• Alternative Catalog Number: BYT-ORB1707717-1,BYT-ORB1707717-10,BYT-ORB1707717-2,BYT-ORB1707717-25,BYT-ORB1707717-5,BYT-ORB1707717-50
• Manufacturer: Biorbyt
• Category: Biochemikalien
• Alternative Names: Cav1.2, Cav3.1, Cav3.2, Cav3.3, ACT 709478, ACT709478, ACT-709478, NBI827104, NBI 827104

Product Description

Apinocaltamide (ACT-709478) is a brain-penetrant, selective T-type calcium channel blocker with IC50 values of 6.4-18 nM against Cav3.1, Cav3.2, and Cav3.3 subtypes. This compound is a valuable research tool for investigating epilepsy and related neurological disorders in both in vitro and in vivo experimental models.

Product Properties

• Molecular Weight: 425.41
• Purity: 99.80% (May vary between batches)
• CAS Number: [1838651-58-3]
• Formula: C22H18F3N5O
• Target: Calcium Channel

Application Notes

• Application Notes: Solubility: 10% DMSO+40% PEG300+5% Tween-80+45% Saline:3.3 mg/mL (7.76 mM),DMSO:120 mg/mL (282.08 mM)