J-2156 is a potent and selective somatostatin SST4 receptor agonist, exhibiting IC50 values of 0.05 nM (human) and 0.07 nM (rat). In rat models of neuropathic pain, it alleviates mechanical allodynia and hyperalgesia with ED50 values of 3.7 and 8.0 mg/kg, respectively, supporting its use in pain research.
Molecular Weight:
468.57
CAS Number:
[848647-56-3]
Formula:
C24H28N4O4S
Target:
Others,Somatostatin
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