The Melatonin-Tamoxifen Conjugate (16c) is a dual-acting small molecule that antagonizes ERalpha and binds melatonin MT1 receptors. It demonstrates anticancer activity in vitro, with IC50 values in the low micromolar range against breast and fibrosarcoma cell lines, and modulates beta-arrestin and ERK signaling pathways.
Molecular Weight:
742.99
Formula:
C47H58N4O4
Target:
Melatonin Receptor
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