SBI-810 is a beta-arrestin-biased allosteric modulator of NTSR1. In the presence of neurotensin, it selectively antagonizes Gq and Gi1 signaling while permitting GoA and G12 activation. This tool compound is used in vitro to study biased NTSR1 signaling pathways and receptor pharmacology.
Molecular Weight:
446.59
CAS Number:
[1849603-79-7]
Formula:
C27H34N4O2
Target:
Neurotensin Receptor
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