Azamulin is a selective, irreversible inhibitor of cytochrome P450 (CYP) 3A isoforms (IC50 values range from 26 to 240 nM for CYP3A4 and CYP3A4/5 from different sources).It is at least 50-fold less potent against CYP2J2 and 100-fold less effective against all other CYP isoforms.Azamulin potently blocks the hydroxylation of testosterone and midazolam by CYP3A4.
Molecular Weight:
478.65
CAS Number:
[76530-44-4]
Formula:
C24H38N4O4S
Target:
Cytochromes P450
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