1-Azakenpaullone, CAS [[676596-65-9]]

Product Overview

• Article Name: 1-Azakenpaullone, CAS [[676596-65-9]]
• Biozol Catalog Number: ENZ-ALX-270-430-M005
• Supplier Catalog Number: ALX-270-430-M005
• Alternative Catalog Number: ENZ-ALX-270-430-M005-5
• Manufacturer: Enzo Life Sciences
• Category: Biochemikalien
• Alternative Names: 9-Bromo-7,12-dihydropyrido[3,2:2,3]azepino[4,5-b]indol-6(5H)-one, 1-AKP

Product Description

Analog of kenpaullone (Prod. No. BML-EI310) acting as a potent and ATP-competitive inhibitor of GSK-3beta (IC50=18nM). Displays ~100-200 fold greater selectivity on GSK-3beta than over CDK1/cyclin B and CDK5/p25 (IC50=2.0µM and 4.2µM, respectively).

Product Properties

• Molecular Weight: 328.2
• Purity: 95% (HPLC, TLC)
• CAS Number: [676596-65-9]
• Formula: C15H10BrN3O
• Target: GSK-3beta