Very potent allosteric modulator of muscarinic receptors, selective for M2-receptors. Retards the dissociation of the antagonist N-methylscopolamine. Affinity for the free receptor is about 10-fold higher than with W84 (Prod. No. ALX-550-399). pKA=7.08,
Molecular Weight:
736.6
Purity:
98% (HPLC)
CAS Number:
[402475-33-6]
Formula:
C34H48Br2N4O4
Target:
Muscarinic acetylcholine receptor M2
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